Discovery of [Cis-3-({(5r)5-[(7-Fluoro-1,1-Dimethyl-2,3-Dihydro1Hinden-5-Yl)carbamoyl]-2-Methoxy-7,8-Dihydro-1,6-Naphthyridin-6(5H)yl}carbonyl)cyclobutyl]acetic Acid (TAK-828F) as a Potent, Selective, and Orally Available Novel Retinoic Acid Receptor-Related Orphan Receptor T Inverse Agonist

doi 10.1021/acs.jmedchem.8b00061.s002
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American Chemical Society (ACS)


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