N-(5-Chloro-1, 3-Benzodioxol-4-Yl)-7-[2-(4-Methylpiperazin-1-Yl)ethoxy]-5-(Tetrahydro-2h-Pyran-4-Yloxy)quinazolin-4-Amine, a Novel, Highly Selective, Orally Available, Dual-Specific C-SRC/Abl Kinase Inhibitor

doi 10.1021/jm060434q.s002
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American Chemical Society (ACS)