Utility of an "Allosteric Site-Impaired" M2 Muscarinic Acetylcholine Receptor as a Novel Construct for Validating Mechanisms of Action of Synthetic and Putative Endogenous Allosteric Modulators

Molecular Pharmacology - United States
doi 10.1124/mol.118.112490
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American Society for Pharmacology & Experimental Therapeutics (ASPET)

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