The Predicted 3D Structure of the Human D2 Dopamine Receptor and the Binding Site and Binding Affinities for Agonists and Antagonists

Proceedings of the National Academy of Sciences of the United States of America - United States
doi 10.1073/pnas.0400100101
Full Text
Abstract

Available in full text

Date
Authors
Publisher

Proceedings of the National Academy of Sciences

Related search

Analogues of the Dopamine D2 Receptor Antagonist L741,626: Binding, Function, and SAR

Bioorganic and Medicinal Chemistry Letters
Organic ChemistryMolecular MedicineMolecular BiologyBiochemistryClinical BiochemistryPharmaceutical ScienceDrug Discovery
2007English

Binding Modes of Full and Partial Agonists in the Orthosteric Binding Site of the Glycine Receptor

Biophysical Journal
Biophysics
2017English

Hydrophobic Residues of the D2 Dopamine Receptor Are Important for Binding and Signal Transduction

Journal of Neurochemistry
BiochemistryMolecular NeuroscienceCellular
2002English

Cannabinoid Agonists and Antagonists Discriminated by Receptor Binding in Rat Cerebellum

British Journal of Pharmacology
Pharmacology
1999English

A Cysteine Residue in the Third Membrane-Spanning Segment of the Human D2 Dopamine Receptor Is Exposed in the Binding-Site Crevice.

Proceedings of the National Academy of Sciences of the United States of America
Multidisciplinary
1994English

Yawning and Hypothermia in Rats: Effects of Dopamine D3 and D2 Agonists and Antagonists

Psychopharmacology
Pharmacology
2007English

Localization of Dopamine D2 Receptor mRNA and D1 and D2 Receptor Binding in the Rat Brain and Pituitary: An in Situ Hybridization- Receptor Autoradiographic Analysis

Journal of Neuroscience
Neuroscience
1990English

Direct Measurements of VEGF:VEGFR2 Binding Affinities Reveal the Coupling Between Ligand Binding and Receptor Dimerization

Journal of Biological Chemistry
BiochemistryCell BiologyMolecular Biology
2019English

Novel and Potent Dopamine D2 Receptor (D2R) Go-Protein Biased Agonists

ACS Pharmacology & Translational Science
2019English

Amanote Research

Note-taking for researchers

Follow Amanote

© 2024 Amaplex Software S.P.R.L. All rights reserved.

Privacy PolicyRefund Policy