Discovery of Clinical Candidate (1R,4r)4-((R)2-((S)6-Fluoro5Himidazo[5,1a]isoindol-5-Yl)-1-Hydroxyethyl)cyclohexan-1-Ol (Navoximod) a Potent and Selective Inhibitor of Indoleamine 2,3-Dioxygenase 1

doi 10.1021/acs.jmedchem.9b00662.s001
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American Chemical Society (ACS)


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