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4, 5-Dihydroxypyrimidine Carboxamides and N-Alkyl-5-Hydroxypyrimidinone Carboxamides Are Potent, Selective HIV Integrase Inhibitors With Good Pharmacokinetic Profiles in Preclinical Species
doi 10.1021/jm060854f.s001
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American Chemical Society (ACS)
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