Structure–Activity Relationships of Peptides Incorporating a Bioactive Reverse-Turn Heterocycle at the Melanocortin Receptors: Identification of a 5800-Fold Mouse Melanocortin-3 Receptor (mMC3R) Selective Antagonist/Partial Agonist Versus the Mouse Melanocortin-4 Receptor (mMC4R)

Journal of Medicinal Chemistry - United States
doi 10.1021/jm301253y
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American Chemical Society (ACS)

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