Discover open access scientific publications

Search, annotate, share and cite publications

Publications by Bjorn R. van Doodewaerd

The Alkyne Moiety as a Latent Electrophile in Irreversible Covalent Small Molecule Inhibitors of Cathepsin K

Journal of the American Chemical Society

Surface Chemistry

English

Related publications

The Nitro Group as a Masked Electrophile in Covalent Enzyme Inhibition

English

Structural Basis of ALDH1A2 Inhibition by Irreversible and Reversible Small Molecule Inhibitors

English

Discovery of the First Irreversible Small Molecule Inhibitors of the Interaction Between the Vitamin D Receptor and Coactivators

Journal of Medicinal Chemistry

Molecular Medicine

English

Identification of Small Molecule Enzyme Inhibitors as Broad-Spectrum Anthelmintics

Scientific Reports

Multidisciplinary

English

Privileged Electrophile Sensors: A Resource for Covalent Drug Development

Cell Chemical Biology

Molecular Medicine

Molecular Biology

Clinical Biochemistry

English

Small Molecule Inhibitors of Metabolic Enzymes Repurposed as a New Class of Anthelmintics

ACS Infectious Diseases

Infectious Diseases

English

Small Molecule Inhibitors of Metabolic Enzymes Repurposed as a New Class of Anthelmintics

English

Small-Molecule Inhibitors of the PI3K Signaling Network

Future Medicinal Chemistry

Molecular Medicine

English

High-Throughput Mass Spectrometric Analysis of Covalent Protein-Inhibitor Adducts for the Discovery of Irreversible Inhibitors

Journal of Biomolecular Screening

Molecular Medicine

Analytical Chemistry

English