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Publications by Kalapala Venkateswara Rao

Novel P2 Tris-Tetrahydrofuran Group in Antiviral Compound1(GRL-0519) Fills the S2 Binding Pocket of Selected Mutants of HIV-1 Protease

Journal of Medicinal Chemistry

Drug Discovery

Molecular Medicine

2013

English

Halogen Bond Interactions of Novel HIV-1 Protease Inhibitors (PI)(GRL-001-15 and GRL-003-15) With the Flap of Protease Are Critical for Their Potent Activity Against Wild-Type and Multi-Pi-Resistant HIV-1 Variants

Antimicrobial Agents and Chemotherapy

Infectious Diseases

Pharmacology

2019

English

Related publications

482 GRL-142, a Novel HIV-1 Protease Inhibitor, Potently Blocks HIV-1 Ex Vivo Infection of Langerhans Cells Within Epithelium

Journal of Investigative Dermatology

English

HIV-1 Protease Dimerization Dynamics Reveals a Transient Druggable Binding Pocket at the Interface

Scientific Reports

Multidisciplinary

2015

English

Targeting Structural Flexibility in HIV-1 Protease Inhibitor Binding

English

Novel Protease Inhibitors Containing C-5-Modified Bis-THF and Aminobenzothiazole as P2 and P2′ Ligands That Exert Potent Antiviral Activity Against Highly Multidrug-Resistant HIV-1 With High Genetic Barrier Against the Emergence of Drug Resistance.

Antimicrobial Agents and Chemotherapy

Infectious Diseases

Pharmacology

2019

English

Understanding HIV-1 Protease Autoprocessing for Novel Therapeutic Development

Future Medicinal Chemistry

English

GS-8374, a Prototype Phosphonate-Containing Inhibitor of HIV-1 Protease, Effectively Inhibits Protease Mutants With Amino Acid Insertions

English

Association of Patient Out-Of-Pocket Costs With Prescription Abandonment and Delay in Fills of Novel Oral Anticancer Agents

Journal of Clinical Oncology

English

Interactions of a Novel Inhibitor From an ExtremophilicBacillussp. With HIV-1 Protease

Journal of Biological Chemistry

English

Amanote Research

Discover open access scientific publications

Search, annotate, share and cite publications

Publications by Kalapala Venkateswara Rao

Novel P2 Tris-Tetrahydrofuran Group in Antiviral Compound1(GRL-0519) Fills the S2 Binding Pocket of Selected Mutants of HIV-1 Protease

Halogen Bond Interactions of Novel HIV-1 Protease Inhibitors (PI)(GRL-001-15 and GRL-003-15) With the Flap of Protease Are Critical for Their Potent Activity Against Wild-Type and Multi-Pi-Resistant HIV-1 Variants

Related publications

482 GRL-142, a Novel HIV-1 Protease Inhibitor, Potently Blocks HIV-1 Ex Vivo Infection of Langerhans Cells Within Epithelium

HIV-1 Protease Dimerization Dynamics Reveals a Transient Druggable Binding Pocket at the Interface

Targeting Structural Flexibility in HIV-1 Protease Inhibitor Binding

Novel Protease Inhibitors Containing C-5-Modified Bis-THF and Aminobenzothiazole as P2 and P2′ Ligands That Exert Potent Antiviral Activity Against Highly Multidrug-Resistant HIV-1 With High Genetic Barrier Against the Emergence of Drug Resistance.

Understanding HIV-1 Protease Autoprocessing for Novel Therapeutic Development

GS-8374, a Prototype Phosphonate-Containing Inhibitor of HIV-1 Protease, Effectively Inhibits Protease Mutants With Amino Acid Insertions

Association of Patient Out-Of-Pocket Costs With Prescription Abandonment and Delay in Fills of Novel Oral Anticancer Agents

Interactions of a Novel Inhibitor From an ExtremophilicBacillussp. With HIV-1 Protease