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Publications by Rita Scarpelli

Discovery of a New Class of Highly Potent Inhibitors of Acid Ceramidase: Synthesis and Structure–Activity Relationship (SAR)

Journal of Medicinal Chemistry

Drug Discovery

Molecular Medicine

2013

English

Structural Determinants of Peripheral O-Arylcarbamate FAAH Inhibitors Render Them Dual Substrates for Abcb1 and Abcg2 and Restrict Their Access to the Brain

Pharmacological Research

Pharmacology

2014

English

Related publications

Discovery and Refinement of a New Structural Class of Potent Peptide Deformylase Inhibitors

English

Discovery of Aminoquinazolines as Potent, Orally Bioavailable Inhibitors of Lymphocyte-Specific Kinase: Synthesis, Structure-Activity Relationship, and in Vivo Anti-Inflammatory Activity

English

Benzoxazolone Carboxamides: Potent and Systemically Active Inhibitors of Intracellular Acid Ceramidase

Angewandte Chemie - International Edition

Catalysis

Chemistry

2014

English

Benzoxazolone Carboxamides: Potent and Systemically Active Inhibitors of Intracellular Acid Ceramidase

Angewandte Chemie - International Edition

Catalysis

Chemistry

2014

English

Structure-Activity Relationship of Potent Photo-Switchable Neuromuscular Inhibitors

Biophysical Journal

Biophysics

2019

English

Highly Selective and Potent Human Β-Secretase 2 (BACE2) Inhibitors Against Type 2 Diabetes: Design, Synthesis, X-Ray Structure and Structure-Activity Relationship Studies

English

Discovery, Synthesis, and in Vivo Activity of a New Class of Pyrazoloquinazolines as Selective Inhibitors of Aurora B Kinase

English

Design, Synthesis and Structure–activity Relationship (SAR) Studies of 2,4-Disubstituted Pyrimidine Derivatives: Dual Activity as Cholinesterase and Aβ-Aggregation Inhibitors

Bioorganic and Medicinal Chemistry

Clinical Biochemistry

Pharmaceutical Science

Drug Discovery

2011

English

Angiotensin-Converting Enzyme Inhibitors: Synthesis and Structure-Activity Relationships of Potent N-Benzyloxycarbonyl Tripeptide Inhibitors.

Chemical and Pharmaceutical Bulletin

English

Amanote Research

Discover open access scientific publications

Search, annotate, share and cite publications

Publications by Rita Scarpelli

Discovery of a New Class of Highly Potent Inhibitors of Acid Ceramidase: Synthesis and Structure–Activity Relationship (SAR)

Structural Determinants of Peripheral O-Arylcarbamate FAAH Inhibitors Render Them Dual Substrates for Abcb1 and Abcg2 and Restrict Their Access to the Brain

Related publications

Discovery and Refinement of a New Structural Class of Potent Peptide Deformylase Inhibitors

Discovery of Aminoquinazolines as Potent, Orally Bioavailable Inhibitors of Lymphocyte-Specific Kinase: Synthesis, Structure-Activity Relationship, and in Vivo Anti-Inflammatory Activity

Benzoxazolone Carboxamides: Potent and Systemically Active Inhibitors of Intracellular Acid Ceramidase

Benzoxazolone Carboxamides: Potent and Systemically Active Inhibitors of Intracellular Acid Ceramidase

Structure-Activity Relationship of Potent Photo-Switchable Neuromuscular Inhibitors

Highly Selective and Potent Human Β-Secretase 2 (BACE2) Inhibitors Against Type 2 Diabetes: Design, Synthesis, X-Ray Structure and Structure-Activity Relationship Studies

Discovery, Synthesis, and in Vivo Activity of a New Class of Pyrazoloquinazolines as Selective Inhibitors of Aurora B Kinase

Design, Synthesis and Structure–activity Relationship (SAR) Studies of 2,4-Disubstituted Pyrimidine Derivatives: Dual Activity as Cholinesterase and Aβ-Aggregation Inhibitors

Angiotensin-Converting Enzyme Inhibitors: Synthesis and Structure-Activity Relationships of Potent N-Benzyloxycarbonyl Tripeptide Inhibitors.