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Publications by Yves Leblanc

Identification of a Benzoisoxazoloazepine Inhibitor (CPI-0610) of the Bromodomain and Extra-Terminal (BET) Family as a Candidate for Human Clinical Trials

Journal of Medicinal Chemistry

Drug Discovery

Molecular Medicine

2016

English

Conformation-Assisted Inhibition of Protein-Tyrosine Phosphatase-1b Elicits Inhibitor Selectivity Over T-Cell Protein-Tyrosine Phosphatase

Journal of Biological Chemistry

English

Related publications

Exploring Selective Inhibition of the First Bromodomain of the Human Bromodomain and Extra-Terminal Domain (BET) Proteins

English

Suppression of Interferon Β Gene Transcription by Inhibitors of Bromodomain and Extra-Terminal (BET) Family Members

English

Inhibition of Bromodomain and Extra-Terminal Proteins (BET) as a Potential Therapeutic Approach in Haematological Malignancies: Emerging Preclinical and Clinical Evidence

Therapeutic Advances in Hematology

Hematology

2015

English

Preclinical Evaluation of the BET Bromodomain Inhibitor BAY 1238097 for the Treatment of Lymphoma

British Journal of Haematology

Hematology

2017

English

The Bromodomain BET Inhibitor JQ1 Suppresses Tumor Angiogenesis in Models of Childhood Sarcoma

Molecular Cancer Therapeutics

Cancer Research

Oncology

2016

English

Identification of a Potent, Highly Selective, and Brain Penetrant Phosphodiesterase 2A Inhibitor Clinical Candidate

English

Bromodomain and Extra-Terminal Protein Inhibition Attenuates Neutrophil-Dominant Allergic Airway Disease

Scientific Reports

Multidisciplinary

2017

English

Identification of Haptoglobin as a Natural Inhibitor of Trypanocidal Activity in Human Serum.

Proceedings of the National Academy of Sciences of the United States of America

Multidisciplinary

1995

English

BET Protein Bromodomain Inhibitor-Based Combinations Are Highly Active Against Post-Myeloproliferative Neoplasm Secondary AML Cells

English

Amanote Research

Discover open access scientific publications

Search, annotate, share and cite publications

Publications by Yves Leblanc

Identification of a Benzoisoxazoloazepine Inhibitor (CPI-0610) of the Bromodomain and Extra-Terminal (BET) Family as a Candidate for Human Clinical Trials

Conformation-Assisted Inhibition of Protein-Tyrosine Phosphatase-1b Elicits Inhibitor Selectivity Over T-Cell Protein-Tyrosine Phosphatase

Related publications

Exploring Selective Inhibition of the First Bromodomain of the Human Bromodomain and Extra-Terminal Domain (BET) Proteins

Suppression of Interferon Β Gene Transcription by Inhibitors of Bromodomain and Extra-Terminal (BET) Family Members

Inhibition of Bromodomain and Extra-Terminal Proteins (BET) as a Potential Therapeutic Approach in Haematological Malignancies: Emerging Preclinical and Clinical Evidence

Preclinical Evaluation of the BET Bromodomain Inhibitor BAY 1238097 for the Treatment of Lymphoma

The Bromodomain BET Inhibitor JQ1 Suppresses Tumor Angiogenesis in Models of Childhood Sarcoma

Identification of a Potent, Highly Selective, and Brain Penetrant Phosphodiesterase 2A Inhibitor Clinical Candidate

Bromodomain and Extra-Terminal Protein Inhibition Attenuates Neutrophil-Dominant Allergic Airway Disease

Identification of Haptoglobin as a Natural Inhibitor of Trypanocidal Activity in Human Serum.

BET Protein Bromodomain Inhibitor-Based Combinations Are Highly Active Against Post-Myeloproliferative Neoplasm Secondary AML Cells