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Publications in Drug Discovery
Quinoline-Based Imidazole-Fused Heterocycles as New Inhibitors of 15-Lipoxygenase
Journal of Enzyme Inhibition and Medicinal Chemistry
Medicine
Drug Discovery
Pharmacology
Plasmatic Exosomes From Prostate Cancer Patients Show Increased Carbonic Anhydrase IX Expression and Activity and Low pH
Journal of Enzyme Inhibition and Medicinal Chemistry
Medicine
Drug Discovery
Pharmacology
Evaluation of the Paraoxonase-1 Kinetic Parameters of the Lactonase Activity by Nonlinear Fit of Progress Curves
Journal of Enzyme Inhibition and Medicinal Chemistry
Medicine
Drug Discovery
Pharmacology
Leishmania Infantum Arginase: Biochemical Characterization and Inhibition by Naturally Occurring Phenolic Substances
Journal of Enzyme Inhibition and Medicinal Chemistry
Medicine
Drug Discovery
Pharmacology
Novel Phthalimide Based Analogues: Design, Synthesis, Biological Evaluation, and Molecular Docking Studies
Journal of Enzyme Inhibition and Medicinal Chemistry
Medicine
Drug Discovery
Pharmacology
1D NMR WaterLOGSY as an Efficient Method for Fragment-Based Lead Discovery
Journal of Enzyme Inhibition and Medicinal Chemistry
Medicine
Drug Discovery
Pharmacology
Synthesis and Biological Evaluation of Novel 8-Substituted Quinoline-2-Carboxamides as Carbonic Anhydrase Inhibitors
Journal of Enzyme Inhibition and Medicinal Chemistry
Medicine
Drug Discovery
Pharmacology
Synthesis, Crystal Structure Determination, Biological Screening and Docking Studies of N 1 -Substituted Derivatives of 2,3-Dihydroquinazolin-4(1 H )-One as Inhibitors of Cholinesterases
Bioorganic Chemistry
Organic Chemistry
Biochemistry
Drug Discovery
Molecular Biology
Liquid Chromatography–tandem Mass Spectrometric Assay for the Quantitation in Human Plasma of the Novel Indenoisoquinoline Topoisomerase I Inhibitors, NSC 743400 and NSC 725776
Journal of Pharmaceutical and Biomedical Analysis
Clinical Biochemistry
Drug Discovery
Analytical Chemistry
Spectroscopy
Pharmaceutical Science
Effect of 6-Benzoyl-Benzothiazol-2-One Scaffold on the Pharmacological Profile of Α-Alkoxyphenylpropionic Acid Derived PPAR Agonists
Journal of Enzyme Inhibition and Medicinal Chemistry
Medicine
Drug Discovery
Pharmacology
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