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Publications in Drug Discovery

Structure-Based Design, Synthesis, Evaluation, and Crystallographic Studies of Conformationally Constrained Smac Mimetics as Inhibitors of the X-Linked Inhibitor of Apoptosis Protein (XIAP)†

Journal of Medicinal Chemistry

Drug Discovery

Molecular Medicine

2008

English

Further Studies on Lead Compounds Containing the Opioid Pharmacophore DMT-Tic

Journal of Medicinal Chemistry

Drug Discovery

Molecular Medicine

2008

English

Pyrogallol-Based Molecules as Potent Inhibitors of the Antiapoptotic BCL-2 Proteins

Journal of Medicinal Chemistry

Drug Discovery

Molecular Medicine

2007

English

L337H Mutant of Rat Neuronal Nitric Oxide Synthase Resembles Human Neuronal Nitric Oxide Synthase Toward Inhibitors

Journal of Medicinal Chemistry

Drug Discovery

Molecular Medicine

2009

English

Defunctionalized Lobeline Analogues: Structure−Activity of Novel Ligands for the Vesicular Monoamine Transporter

Journal of Medicinal Chemistry

Drug Discovery

Molecular Medicine

2005

English

New Tacrine−Huperzine a Hybrids (Huprines): Highly Potent Tight-Binding Acetylcholinesterase Inhibitors of Interest for the Treatment of Alzheimer's Disease

Journal of Medicinal Chemistry

Drug Discovery

Molecular Medicine

2000

English

On the Applicability of GPCR Homology Models to Computer-Aided Drug Discovery: A Comparison Between in Silico and Crystal Structures of the Β2-Adrenergic Receptor

Journal of Medicinal Chemistry

Drug Discovery

Molecular Medicine

2008

English

A Comparison of the Binding Sites of Matrix Metalloproteinases and Tumor Necrosis Factor-Α Converting Enzyme: Implications for Selectivity

Journal of Medicinal Chemistry

Drug Discovery

Molecular Medicine

2005

English

Synthesis and Biological Evaluation of Cyclopropyl Analogues of Fosmidomycin as PotentPlasmodiumfalciparumGrowth Inhibitors

Journal of Medicinal Chemistry

Drug Discovery

Molecular Medicine

2006

English

Interactions Between Human Glutamate Carboxypeptidase II and Urea-Based Inhibitors: Structural Characterization†

Journal of Medicinal Chemistry

Drug Discovery

Molecular Medicine

2008

English

Amanote Research

Discover open access scientific publications

Search, annotate, share and cite publications

Publications in Drug Discovery

Structure-Based Design, Synthesis, Evaluation, and Crystallographic Studies of Conformationally Constrained Smac Mimetics as Inhibitors of the X-Linked Inhibitor of Apoptosis Protein (XIAP)†

Further Studies on Lead Compounds Containing the Opioid Pharmacophore DMT-Tic

Pyrogallol-Based Molecules as Potent Inhibitors of the Antiapoptotic BCL-2 Proteins

L337H Mutant of Rat Neuronal Nitric Oxide Synthase Resembles Human Neuronal Nitric Oxide Synthase Toward Inhibitors

Defunctionalized Lobeline Analogues: Structure−Activity of Novel Ligands for the Vesicular Monoamine Transporter

New Tacrine−Huperzine a Hybrids (Huprines): Highly Potent Tight-Binding Acetylcholinesterase Inhibitors of Interest for the Treatment of Alzheimer's Disease

On the Applicability of GPCR Homology Models to Computer-Aided Drug Discovery: A Comparison Between in Silico and Crystal Structures of the Β2-Adrenergic Receptor

A Comparison of the Binding Sites of Matrix Metalloproteinases and Tumor Necrosis Factor-Α Converting Enzyme: Implications for Selectivity

Synthesis and Biological Evaluation of Cyclopropyl Analogues of Fosmidomycin as PotentPlasmodiumfalciparumGrowth Inhibitors

Interactions Between Human Glutamate Carboxypeptidase II and Urea-Based Inhibitors: Structural Characterization†