(PDF) Comparison of the Binding of 3-Flu

Comparison of the Binding of 3-Fluoromethyl-7-Sulfonyl-1, 2, 3, 4-Tetrahydroisoquinolines With Their Isosteric Sulfonamides to the Active Site of Phenylethanolamine N-Methyltransferase1

doi 10.1021/jm060466d.s001

Full Text

Open PDF

Abstract

Available in full text

Date

Unknown

Authors

Unknown

Publisher

American Chemical Society (ACS)

Related search

Studies on Tetrahydroisoquinolines. IV. Synthesis of 4-Alkyl (Phenyl) Amino-7-Hydroxy-6-Methoxy-2-Methyl-1, 2, 3, 4-Tetrahydroisoquinolines

Chemical and Pharmaceutical Bulletin

English

N-[(2-Chlorophenyl)sulfonyl]-3-Nitrobenzamide

Acta Crystallographica Section E Structure Reports Online

2013

English

3-[(4-Fluorophenyl)sulfonyl]-5-Iodo-2-Methyl-1-Benzofuran

Acta Crystallographica Section E Structure Reports Online

2010

English

Studies on Nitrogen-Containing Heterocyclic Compounds. XXXV. Syntheses and Reduction of 4-Amino-2-Cyano-1, 3-Dimethoxy-1, 2, 3, 4-Tetrahydroisoquinolines

Yakugaku Zasshi

Pharmacology

Pharmaceutical Science

1979

English

Exploring the Active Site of Phenylethanolamine N-Methyltransferase With 1,2,3,4-Tetrahydrobenz[h]isoquinoline Inhibitors☆

Bioorganic and Medicinal Chemistry

Clinical Biochemistry

Pharmaceutical Science

Drug Discovery

2007

English

Synthesis of 1-(N-Benzyl-2-Oxo-5-Ethyl-4-Piperidylmethyl)- 6, 7-Dimethoxy-3, 4-Dihydroisoquinoline

Proceedings of the Japan Academy

1954

English

Contributions to N‐2‐4, N‐3‐4, N‐4‐4, Θ‐2‐4, and Θ‐3‐4 Hemispheric Sound Reproduction Technology

Journal of the Acoustical Society of America

English

4-Oxo-1, 2, 3, 4-Tetrahydroquinazoline. IV. Reactions of 2-Chloromethyl-3-Aryl-4-Oxo-1, 2, 3, 4-Tetrahydroquinazolines

Chemical and Pharmaceutical Bulletin

English

Application of the Goldilocks Effect to the Design of Potent and Selective Inhibitors of Phenylethanolamine N-Methyltransferase: Balancing pKa and Steric Effects in the Optimization of 3-Methyl-1, 2, 3, 4-Tetrahydroisoquinoline Inhibitors by B-Fluorination

English

Amanote Research

Comparison of the Binding of 3-Fluoromethyl-7-Sulfonyl-1, 2, 3, 4-Tetrahydroisoquinolines With Their Isosteric Sulfonamides to the Active Site of Phenylethanolamine N-Methyltransferase1

doi 10.1021/jm060466d.s001

Full Text

Abstract

Date

Authors

Publisher

Related search

Studies on Tetrahydroisoquinolines. IV. Synthesis of 4-Alkyl (Phenyl) Amino-7-Hydroxy-6-Methoxy-2-Methyl-1, 2, 3, 4-Tetrahydroisoquinolines

N-[(2-Chlorophenyl)sulfonyl]-3-Nitrobenzamide

3-[(4-Fluorophenyl)sulfonyl]-5-Iodo-2-Methyl-1-Benzofuran

Studies on Nitrogen-Containing Heterocyclic Compounds. XXXV. Syntheses and Reduction of 4-Amino-2-Cyano-1, 3-Dimethoxy-1, 2, 3, 4-Tetrahydroisoquinolines

Exploring the Active Site of Phenylethanolamine N-Methyltransferase With 1,2,3,4-Tetrahydrobenz[h]isoquinoline Inhibitors☆

Synthesis of 1-(N-Benzyl-2-Oxo-5-Ethyl-4-Piperidylmethyl)- 6, 7-Dimethoxy-3, 4-Dihydroisoquinoline

Contributions to N‐2‐4, N‐3‐4, N‐4‐4, Θ‐2‐4, and Θ‐3‐4 Hemispheric Sound Reproduction Technology

4-Oxo-1, 2, 3, 4-Tetrahydroquinazoline. IV. Reactions of 2-Chloromethyl-3-Aryl-4-Oxo-1, 2, 3, 4-Tetrahydroquinazolines

Application of the Goldilocks Effect to the Design of Potent and Selective Inhibitors of Phenylethanolamine N-Methyltransferase: Balancing pKa and Steric Effects in the Optimization of 3-Methyl-1, 2, 3, 4-Tetrahydroisoquinoline Inhibitors by B-Fluorination